It is a psychoactive compound with nootropic and tranquilizing effects. It was initially synthesized in Russia during the 1960s. It is a derivative of the neurotransmitter gamma-aminobutyric acid (GABA). It was designed to cross the blood-brain barrier more effectively than GABA itself.
Phenibut HCl for sale mimics GABA’s inhibitory effects. It offers relief from anxiety, stress, and sleep disturbances. It holds promise for enhancing cognitive function and reducing anxiety.
Let’s explore gaba derivative Phenibut in depth in this article. We’ll cover its mechanisms of action, benefits, dosages, safety considerations, and where to buy it.
What is Phenibut HCl?
- CAS Number is stated as 1078-21-3
- Molar Mass is 179.219 g·mol−1
- It has a Chemical Formula of C10H13NO2
- IUPAC Name is 4-Amino-3-phenylbutanoic acid
- Also known by Synonyms as Amino phenylbutyric acid; Fenibut; Fenigam; Phenigam; Phenybut; Phenygam; Phenylgamma; Phenigama; PHG; PhGABA; β-Phenyl-γ-aminobutyric acid; β-Phenyl-GABA, GABA-derivative phenibut
It is a modified form of GABA, known as β-phenyl-GABA, which is more easily absorbed by the brain. It acts primarily as a GABA receptor agonist phenibut. It is similar to the drug baclofen, which promotes relaxation, reduces anxiety, and improves sleep quality.
Phenibut HCl is also believed to modulate dopamine levels. This contributes to its mood-enhancing properties.
It was originally developed in Russia. Phenibut was used as a non-addictive alternative to other psychoactive drugs. It is not approved by the FDA for medical use in the United States.
How Does Phenibut HCl Work?
It works by binding to GABA-B receptors in the brain. These are part of the GABAergic system. These are responsible for reducing neuronal excitability and promoting a calming effect. By mimicking GABA, Phenibut helps to inhibit excessive neural activity. This leads to reduced anxiety, enhanced relaxation, and improved sleep.
Also, Phenibut’s ability to cross the blood-brain barrier is facilitated by its chemical structure. It is specifically because of the addition of a phenyl ring. This structural modification allows Phenibut to enter the brain more effectively than GABA.
Once inside the brain, it exerts its effects on GABA-B receptors. It may also interact with dopamine receptors, which could explain its mood-enhancing properties.
Phenibut’s effects typically begin within 2 to 4 hours after ingestion. Its peak effects occur around 4 to 6 hours. These effects last for several hours. Therefore, it is effective for temporary relief from anxiety and stress.
Benefits of Phenibut HCl
Below are some of the primary benefits associated with Phenibut HCl:
Anxiety and Stress Reduction
Phenibut HCl is widely recognized for its anxiolytic properties. Activating GABA-B receptors helps calm the nervous system. It also reduces feelings of anxiety and stress. This is useful for individuals dealing with social anxiety or performance anxiety. [R]
Improved Sleep Quality
Phenibut HCl’s calming effects extend to sleep. It helps improve both the quality and duration of sleep. It is often used to treat insomnia and other sleep disorders. It promotes deeper and more restful sleep. [R]
Cognitive Enhancement
As a nootropic drug, Phenibut HCl has been reported to enhance cognitive functions. This includes memory, focus, and learning. Its ability to reduce anxiety may contribute to improved cognitive performance. Since it alleviates stress-related cognitive impairments. [R]
Mood Enhancement
Phenibut nootropic modulates dopamine levels. It elevates mood and alleviates symptoms of mild depression. Users often report feelings of well-being and increased sociability after taking Phenibut. [R]
Relief from Withdrawal Symptoms
Phenibut HCl is sometimes used to reduce withdrawal symptoms. Usually from substances like alcohol and benzodiazepines. Its effects on the GABAergic system help to reduce the severity of withdrawal symptoms. [R]
This makes it easier for individuals to manage their recovery.
How to Take Phenibut HCl
Phenibut HCl is available in various forms, including powder and capsules. The method of administration can influence how quickly and effectively the compound works.
Phenibut HCl Powder
The powder form of Phenibut HCl is versatile. It allows for precise dosage adjustments. It can be mixed with water or juice and is typically taken on an empty stomach to enhance absorption.
Phenibut HCl Capsules
Capsules offer a more convenient way to take Phenibut HCl. Especially for those who prefer not to deal with measuring out powder. Phenibut capsules also help to mask the taste of Phenibut, which can be unpleasant.
Recommended Phenibut Dosage
This varies depending on the intended use and individual tolerance. It’s important to start with a low dose and gradually increase it as needed.
For Anxiety Relief
A typical starting dose is 200-300 mg, taken once or twice per week. This dose helps reduce anxiety without causing significant sedation or other side effects.
For Sleep Improvement
A dose of 500-1000 mg taken in the evening helps to promote relaxation and improve sleep quality. It’s essential to avoid taking Phenibut daily to prevent dependence.
For Cognitive Enhancement
Lower doses of 250-500 mg are often used to enhance focus and cognitive performance. These doses can be taken in the morning or early afternoon.
Avoiding High Doses
Doses above 1500 mg are not recommended, especially for those new to Phenibut. High doses increase the risk of side effects, tolerance, and dependence.
Cycling
Phenibut HCl should not be taken more than twice a week to minimize the risk of dependence. It’s also advisable to cycle off Phenibut after several weeks of use. This will allow the body to reset and reduce the risk of withdrawal symptoms.
Potential Side Effects
- Dependence and Withdrawal
- Fatigue and Sedation
- Nausea and Headaches
- Cognitive Impairment
- Psychiatric Effects
Where to Buy Phenibut Online?
Behemothlabz is a trusted provider of high-quality Phenibut HCl capsules. They offer products that are tested for purity and potency. They provide free shipping on orders over $100. They will ensure that you receive your Phenibut quickly and discreetly.
Behemothlabz stands out as the best source for Phenibut HCl. They do not just offer top-quality products but also excellent customer service. Behemothlabz also offers phenibut FAA or free amino acid. Behemothlabz has you covered.
FAQs
Is Phenibut HCl legal?
The legal status of Phenibut HCl varies by country. In the United States, it is legal to buy and sell Phenibut as a dietary supplement. However, the FDA does not approve it for medical use.
Other countries, like Australia and Canada, have placed restrictions on Phenibut due to safety concerns.
Can Phenibut HCl be taken daily?
No, Phenibut HCl should not be taken daily. Frequent use can lead to tolerance, dependence, and withdrawal symptoms. It’s recommended to limit usage to no more than twice a week and to cycle off periodically.
What are the signs of Phenibut overdose?
These may include extreme drowsiness, confusion, agitation, nausea, vomiting, and loss of coordination. In severe cases, respiratory depression and loss of consciousness can occur. If you suspect an overdose, seek medical attention immediately.
How does Phenibut HCl compare to other nootropics?
Phenibut HCl is unique among nootropics. It is due to its tranquilizing effects and potential for dependence. It can enhance cognitive function by reducing anxiety. But, it carries risks compared to other nootropics like racetams or modafinil.
Can Phenibut HCl help with alcohol withdrawal?
Yes, Phenibut HCl has been used to alleviate symptoms of alcohol withdrawal. This is due to its effects on the GABAergic system.
Conclusion
Phenibut HCl is a powerful GABA derivative with calming and cognitive-enhancing effects. It can help reduce anxiety, improve sleep, and boost mental function.
However, it also comes with serious risks like dependence and withdrawal.
Use Phenibut HCl safely. Follow proper dosage guidelines, cycle your use, and buy from trusted sources like Behemothlabz. If you’re thinking about trying Phenibut HCl, carefully consider the benefits and adverse reactions. Always consult a healthcare professional.