Don’t get confused if you hear the term “Arimistane” for the first time! Arimistane was originally researched for breast cancer treatment in menopausal women. [1] In the context of fitness and bodybuilding, Arimistane is used to block the unwanted or extra estrogens in the body.
In this blog, we’ll give you an insight on what Arimistane is, its mechanism of action, its potential benefits & side effects, and appropriate dosage. We’ll also discuss its uses, and role in bodybuilding.
What is Arimistane?
Arimistane, also referred to as Androsta-3,5-diene-7,17-dione is a non-steroidal compound that leaves the Aromatase enzyme inactive or blocked. Aromatase enzyme converts the testosterone into estrogens. When the Aromatase enzyme is blocked, your body stops converting testosterone into estrogen.
In men, testosterone converts into estrogens through aromatization. However, when the amount of estrogen increases it causes serious problems such as gynecomastia (enlargement of the breast tissue in men), erectile dysfunction, reduced libido, and decreased muscle mass.
Athletes or bodybuilders who use anabolic steroids to gain muscle mass and strength often experience increased estrogen levels. They may turn to Arimistane to boost testosterone and reduce estrogen levels.
How Does Arimistane (Aromatase Inhibitor) Work?
Arimistane works by inhibiting the enzyme aromatase. When the enzyme Aromatase (responsible for converting testosterone into estrogens) is blocked, the amount of estrogen produced in the body is reduced, ultimately leading to balanced hormones. [2]
Potential Benefits of Arimistane for Bodybuilders
Users who have used Arimistane described its potential effects. Some of which we have discussed below:
- Reduces Estrogen Levels
- Increases Testosterone
- Reduces Water Retention
- Improved Mood and Libido
Reduces Estrogen Levels:
One of the primary benefits of Arimistane is that it reduces the estrogen levels. High estrogen levels in men can cause unwanted issues such as water retention, fat gain, and gynecomastia. Decreased estrogen levels can help in balancing hormones, which can lead to enhanced muscle definition. [3]
Increases Testosterone:
When your body detects the lower estrogen levels, it automatically boosts testosterone production. Higher testosterone levels can result in increased muscle mass, and speedy recovery after intense workouts. [4]
Reduces Water Retention:
Higher estrogen levels can cause your body to hold onto excess water, which gives you a bloated appearance. Arimistane gives you a more defined and vascular physique by eliminating water retention. This is particularly beneficial when you are in your cutting phases aiming to achieve a leaner and sharper body.
Improved Mood and Libido:
Bodybuilders who do intense workouts may experience hormone imbalances that could affect their mood and libido. Arimistane (AI) helps boost mood and libido by offering hormonal balance. When you are in a good mood and your mind is clear you can better focus on your workout sessions.[5]
Speedy Recovery and Reducing Muscle Breakdown:
Arimistane keeps estrogen levels in check and helps maintain an anabolic state that reduces muscle catabolism (breakdown). This ensures that bodybuilders can recover easily without wasting muscle mass when they are doing intense workout training.
Furthermore, Arimistane promotes testosterone levels by inhibiting the aromatase enzyme, which allows for faster muscle repair and regeneration.
Potential Side Effects of Arimistane
According to purported reports, Arimistane might have the following side effects:
- Joint Pain
- Fatigue & Mood Swings
- Headaches
- Hot flashes
Before and After Results of Using Arimistane
Various users have used Arimistane to boost testosterone and improve muscle mass. Here are the before and after results of those who have used Arimistane.
Before Using Arimistane
Here are the results users reported before they used Arimistane.
- Increased Estrogen Levels
Users who were not using Arimistane during a steroid or prohormone cycle experienced an increase in estrogen production.
- Water Retention:
Some users might experience elevated estrogen levels due to the conversion of testosterone into estrogen. It causes their body to retain water, leading to a bloated appearance.
- Gynecomastia Risk:
Users also experience enlarged breasts due to increased estrogen levels.
After Using Arimistane
After taking Arimistane the users have reported the following results.
- Reduced Estrogen Levels:
Users experienced reduced estrogen levels after taking Arimistane. Their muscle mass improves as testosterone is boosted.
- Decreased Water Retention:
Many users reported that their physique improved and they got a leaner body. This is because their water retention decreases, leading to less bloating and a more defined shape.
- Decreased Risk of Gynecomastia:
One user, who experienced gynecomastia, reported that it got much better after turning to Arimistane.
Dosage Guidelines and Cycle Length of Arimistane
So far in the blog, you’ve learned what Arimistane is and how it works, including its recommended dosage. Now it’s time for you to find out the dosage and cycle length of Arimistane.
According to users’ experience, Arimistane is used anywhere between 25 mg, 75 mg, 100 mg to 200 mg. You can choose a dosage according to your workout routine. However, we recommend you start from lower doses.
As for post-cycle therapy length, most users have reported using it for roughly 4 to 8 weeks.
Note: To get the most authentic information on dosage and PCT, we recommend you consult with your healthcare provider.
Where To Buy Arimistane?
You can buy Arimistane and other products such as SARMs, peptides, and nootropics, for research purposes from the following vendors:
| Vendors | Price Range | Free Shipping | Verdict | Buying Link |
| Purerawz | $30.98 – $106.98 | Free shipping for orders above $100 | Purerawz has been around for many years and has garnered a good reputation among others for its high quality and standard products. | Buy Arimistane from Purerawz |
| Behemoth Labz | $26.48 – $65.98 | Free shipping on any order over $100 | The online shop offers first and third-party-tested products at affordable prices. | Buy Arimistane from Behemoth Labz |
| Iron Mountain Labz | $92.48 | Free shipping on orders over $150 | This online shop has the best SERMS, Peptides, SARMs, Anabolic, and Kratom. You can order any of the products from this vendor. | Buy Arimistane from Iron Mountain Labz |
Summing Up
Arimistane is used to block the extra estrogen levels. It is important to note that too much testosterone or estrogen is not good for your health. Therefore, you should take estrogen blockers that maintain your hormone levels and help prevent serious problems like gyno and muscle loss.
FAQs
1. When is the Best Time to Take Arimistane?
Many fitness enthusiasts take Arimistane after a cycle of performance enhancers like prohormones. Some also use it after a cycle of SARMS such as Ostarine.
2. Why is Arimistane Used in Bodybuilding?
Bodybuilders who have previously used anabolic steroids and faced issues such as excessive estrogen levels, gynecomastia, and water retention might turn to Arimistane to block all these effects. Arimistane is believed to offer muscle growth without offering side effects often associated with anabolic steroids.
3. How Does Arimistane Treat Gynecomastia In Bodybuilders?
Arimistane may treat gynecomastia by reducing estrogen levels. It inhibits the aromatase enzyme, which is responsible for converting testosterone into estrogen. When the estrogen levels are lower there are minimal chances that bodybuilders encounter gyno.
Arimistane is an effective compound when it comes to treating gynecomastia. Gynecomastia is the condition in which the breast tissue of men gets enlarged. The condition can occur when the estrogen levels in the body are higher. It could happen due to an anabolic steroid cycle.
4. Why do Bodybuilders and Athletes Choose Arimistane?
Bodybuilders and other athletes might use Arimistane to balance their hormone levels and reduce excess estrogen. A majority of athletes and bodybuilders make use of Arimistane as post-cycle therapy to maintain stability.
5. How Long Does Arimistane Remain in the Body?
Arimistane might stay in your body for around 2-3 days. However, a few factors such as metabolism and dosage may influence this timeframe.
Reference
- M, S., & Gl, P. (2008). Anastrozole: A Review of Its Use in Postmenopausal Women With Early-Stage Breast Cancer. Drugs. https://pubmed.ncbi.nlm.nih.gov/18547136/
- Aromatase inhibitor. (2023, January 29). Wikipedia. https://en.wikipedia.org/wiki/Aromatase_inhibitor
- Breast Cancer Prevention: Aromatase Inhibitors. (n.d.). Www.cancer.org. https://www.cancer.org/cancer/types/breast-cancer/risk-and-prevention/aromatase-inhibitors-for-lowering-breast-cancer-risk.html
- ARIMISTANE: Overview, Uses, Side Effects, Precautions, Interactions, Dosing and Reviews. (2018). Webmd.com. https://www.webmd.com/vitamins/ai/ingredientmono-1645/arimistane-%5Bfast-facts%5D
- De Ronde, W., & de Jong, F. H. (2011). Aromatase inhibitors in men: effects and therapeutic options. Reproductive Biology and Endocrinology, 9(1), 93. https://doi.org/10.1186/1477-7827-9-93
